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au:Amaral, Maria C. A.
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1.
Detection of plasma anti-lipopolysaccharide (LPS)antibodies against enterohemorrhagic Escherichia coli(EHEC) in asymptomatic kindergarten teachers fromBuenos Aires province
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Fernandez Brando, Romina J.
; Sacerdoti, Flavia
; Amaral, María M.
; Bernal, Alan M.
; Rocha, Marcelo Da
; Belardo, Marcela
; Alermo, Marina S.
; Ibarra, Cristina A.
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Abstract In Argentina, hemolytic uremic syndrome (HUS) caused by EHEC has the highest incidence in the world. EHEC infection has an endemo-epidemic behavior, causing 20-30% of acute bloody diarrhea syndrome in children under 5 years old. In the period 2016-2020, 272 new cases per year were notified to the National Health Surveillance System. Multiple factors are responsible for HUS incidence in Argentina including person-to-person transmission. In order to detect possible EHEC carriers, we carried out a preliminary study of the frequency of kindergarten teachers with anti-LPS antibodies against the most prevalent EHEC serotypes in Argentina. We analyzed 61 kindergarten teachers from 26 institutions from José C. Paz district, located in the suburban area of Buenos Aires province, Argentina. Fifty-one percent of the plasma samples had antibodies against O157, O145, O121 and O103 LPS: 6.4% of the positive samples had IgM isotype (n=2), 61.3% IgG isotype (n=19) and 32.3% IgM and IgG (n=10). Given that antibodies against LPS antigens are usually short-lived specific IgM detection may indicate a recent infection. In addition, the high percentage of positive samples may indicate a frequent exposure to EHEC strains in the cohort studied, as well as the existence of a large non-symptomatic population of adults carrying pathogenic strains that could contribute to the endemic behavior through person-to-person transmission. The improvement of continuous educational programs in kindergarten institutions could be a mandatory measure to reduce HUS cases not only in Argentina but also globally.
Resumen En Argentina, el síndrome urémico hemolítico causado por Escherichia coli enterohemorrágica (EHEC) tiene la más alta incidencia del mundo. Las infecciones por EHEC tienen un comportamiento endemoepidémico y causan del 20 al 30% de los síndromes de diarrea sanguinolenta en niños menores de 5 años. En el período 2016-2020, se notificaron 272 nuevos casos por año al Sistema de Vigilancia de Salud Nacional. Múltiples factores son responsables de la alta incidencia de SUH en Argentina, incluyendo la transmisión persona-persona. Con el objetivo de detectar posibles portadores asintomáticos de EHEC, realizamos un estudio preliminar de la frecuencia de anticuerpos antilipopolisacáridos contra los serotipos de EHEC más prevalentes en Argentina. El estudio se realizó con muestras de plasma obtenidas de 61 maestras y maestros de jardines de infantes de 26 instituciones del distrito de José C. Paz, localizado en el área suburbana de la provincia de Buenos Aires, Argentina. El 51% de las muestras presentaron anticuerpos contra los serotipos de lipopolisacáridos O157, O145, O121 y O103; el 6,4% de las muestras positivas tuvieron el isotipo IgM (n=2), el 61,3% el isotipo IgG (n=19) y el 32,3% los isotipos IgM e IgG (n=10). Dado que los anticuerpos antilipopolisacáridos presentan usualmente una duración corta, la detección de IgM específica podría indicar una infección reciente. Además, el alto porcentaje de muestras positivas hallado podría indicar una exposición frecuente a las cepas de EHEC en la cohorte estudiada. Asimismo, la gran población de adultos portadores asintomáticos de estas cepas patógenas podría contribuir al comportamiento endémico, a través de la transmisión persona-persona. El perfeccionamiento de programas educacionales continuos en jardines de infantes podría constituir una medida importante para reducir los casos de síndrome urémico hemolítico, no solo en Argentina, sino también en el mundo.
2.
Valorization of Hesperidin from Citrus Residues: Evaluation of Microwave-Assisted Synthesis of Hesperidin-Mg Complex and Their Insecticidal Activity
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Silva, Danielle F. da
; Bomfim, João P. A.
; Marchi, Rafael C.
; Amaral, Jéssica C.
; Pinto, Luciano S.
; Carlos, Rose M.
; Ferreira, Antonio G.
; Forim, Moacir R.
; Fernandes, João B.
; Silva, Maria F. G. F. da
; Oliveira, Regiane C. de
; Buss, David
; Kirk, William D. J.
; Bruce, Toby J. A.
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Journal of the Brazilian Chemical Society
- Métricas do periódico
The aim of the current study was the valorization of hesperidin, the dominant flavonoid in citrus processing waste, by microwave-assisted synthesis of hesperidin-Mg complex, improving its antioxidant activity and insecticidal potential. Here we show, for the first time, that microwave-assisted synthesis of [Mg(hesp)2(phen)]OAc (1) (hesp: hesperidin, phen: phenanthroline) improve the reaction rate and yield. The nuclear magnetic resonance (NMR) experiments proved to be powerful tools for the identification of three isomers in metal complexes. Moreover, we explore the insecticidal potential of 1 and [Mg(phen)2(Isov)]OAc (2) (Isov : isovanillic acid) complexes against three insects. Complex 1 killed 80% of adults whitefly at 0.14 μmol L-1, and 2 76% at 0.36 μmol L-1. There was a total mortality of Spodoptera frugiperda with 2 at 0.39 μmol L-1, and 83% with 1 at 0.14 μmol L-1. Both have similar activity, and represent a novel group of insecticide for Bemisia tabaci and S. frugiperda; nevertheless, the benefits of both as Myzus persicae repellent require further evaluation.
3.
Effective recommendations towards healthy routines to preserve mental health during the COVID-19 pandemic
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Pilz, Luísa K.
; Couto Pereira, Natividade S.
; Francisco, Ana Paula
; Carissimi, Alicia
; Constantino, Débora B.
; Caus, Letícia B.
; Abreu, Ana Carolina O.
; Amando, Guilherme R.
; Bonatto, Fernanda S.
; Carvalho, Paula V.V.
; Cipolla-Neto, José
; Harb, Ana
; Lazzarotto, Gabriela
; Marafiga, Joseane Righes
; Minuzzi, Luciano
; Montagner, Francisco
; Nishino, Fernanda A.
; Oliveira, Melissa A.B.
; dos Santos, Bruno G.T.
; Steibel, Eduardo G.
; Tavares, Patrice S.
; Tonon, André C.
; Xavier, Nicóli B.
; Zanona, Querusche Klippel
; Amaral, Fernanda G.
; Calcagnotto, Maria Elisa
; Frey, Benicio N.
; Hidalgo, Maria Paz
; Idiart, Marco
; Russomano, Thais
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Objective: To assess the adherence to a set of evidence-based recommendations to support mental health during the coronavirus disease 2019 (COVID-19) pandemic and its association with depressive and anxiety symptoms. Methods: A team of health workers and researchers prepared the recommendations, formatted into three volumes (1: COVID-19 prevention; 2: Healthy habits; 3: Biological clock and sleep). Participants were randomized to receive only Volume 1 (control), Volumes 1 and 2, Volumes 1 and 3, or all volumes. We used a convenience sample of Portuguese-speaking participants over age 18 years. An online survey consisting of sociodemographic and behavioral questionnaires and mental health instruments (Patient Health Questionnaire-9 [PHQ-9] and Generalized Anxiety Disorder-7 [GAD-7]) was administered. At 14 and 28 days later, participants were invited to complete follow-up surveys, which also included questions regarding adherence to the recommendations. A total of 409 participants completed the study – mostly young adult women holding university degrees. Results: The set of recommendations contained in Volumes 2 and 3 was effective in protecting mental health, as suggested by significant associations of adherence with PHQ-9 and GAD-7 scores (reflecting anxiety and depression symptoms, respectively). Conclusion: The recommendations developed in this study could be useful to prevent negative mental health effects in the context of the pandemic and beyond.
4.
Design, Synthesis and Anticancer Biological Evaluation of Novel 1,4-Diaryl-1,2,3-triazole Retinoid Analogues of Tamibarotene (AM80)
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Aleixo, Mariana A. A.
; Garcia, Taís M.
; Carvalho, Diego B.
; Viana, Luiz H.
; Amaral, Marcos S.
; Kassab, Najla M.
; Cunha, Marilin C.
; Pereira, Indiara C.
; Guerrero Jr., Palimécio G.
; Perdomo, Renata T.
; Matos, Maria F. C.
; Baroni, Adriano C. M.
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Journal of the Brazilian Chemical Society
- Métricas do periódico
We report herein the design and synthesis via click chemistry of twelve novel triazole retinoid analogues of tamibarotene (AM80) and the evaluation of their anticancer activities against six cancer cell lines: HL60, K562, 786, HT29, MCF7 and PC3. Among the synthesized compounds, two were more potent than tamibarotene against solid tumor cells, and one of them had similar potency to tamibarotene against HL60 cells. The bioisosteric exchange between the amide group and the 1,2,3-triazole core in the retinoid agent tamibarotene (AM80) reported in this work is a valid strategy for the generation of useful compounds against cancer.
https://doi.org/10.21577/0103-5053.20170119
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5.
Antifungal potential of punicalagin against Cryptococcus neoformans species complex
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Silva, Thaísa Cristina
; Zara, Ana Laura de Sene Amâncio
; Sá, Fabyola Amaral da Silva
; Bara, Maria Teresa Freitas
; Ávila, Renato Ivan de
; Costa, Carolina Rodrigues
; Valadares, Marize Campos
; Santos, Andressa Santana dos
; Freitas, Vivianny Aparecida Queiroz
; Silva, Maria do Rosário Rodrigues
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Revista do Instituto de Medicina Tropical de São Paulo
- Métricas do periódico
ABSTRACT This study evaluated the antifungal activity and cytotoxicity profile of the ellagitannin punicalagin, a compound extracted from the L. pacari A. St.-Hil (Lythraceae) leaf, against Cryptococcus neoformans species complex. Minimum inhibitory concentrations (MIC) were checked using the broth microdilution method. Minimum fungicidal concentrations (MFC) and time of death were used to confirm the antifungal activity of the compound. The in vitro cytotoxicity of punicalagin was tested in BALB/c3T3 fibroblasts and A549 human lung cancer cell line, while the hemolytic potential was tested on sheep erythrocytes. The morphological changes induced in yeast strains by the presence of punicalagin were also analyzed. Tested on eight isolates of the C. neoformans complex punicalagin showed MIC of 0.5 to 4.0 μg/mL and MFC> 256 μg/mL. Punicalagin also demonstrated a good growth inhibitory activity in time-kill curves, but it was not able to achieve a statistically significant reduction of fungal growth suggesting a fungistatic effect of the compound. In vitro cytotoxicity studies using the two cell lines showed that punicalagin has low activity on these cells and no activity on sheep erythrocytes. Morphological changes were seen in the yeasts strains studied when treated with punicalagin. Therefore, punicalagin is a potential antifungal for important pathogenic yeasts and presents a low cytotoxicity profile associated with no hemolytic effects.
https://doi.org/10.1590/s1678-9946201860060
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6.
Geo-environmental zoning using physiographic compartmentalization: a proposal for supporting sustainable decision-making
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CORRÊA, CLAUDIA V.S.
; REIS, FÁBIO A.G.V.
; GIORDANO, LUCILIA C.
; BRESSANE, ADRIANO
; CHAVES, CAMILA J.
; AMARAL, ANA MARIA C. DO
; BRITO, HERMES D.
; MEDEIROS, GERSON A. DE
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Anais da Academia Brasileira de Ciências
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ABSTRACT The geo-environmental zoning represents an important strategy in the territorial management. However, it requires a logical and structured procedure. Therefore, an approach using physiographic compartmentalization is proposed and applied as case study in a region covered by the topographic maps of São José dos Campos and Jacareí, Brazil. This region has great geological and geomorphological peculiarities, beyond being a place with large human interventions because of its quickly economic growth. The methodology is based on photointerpretation techniques and remote sensing in GIS environment. As a result, seven geo-environmental zones were obtained from a weighted integration by multicriteria analysis of physiographic units with land-use classes. In conclusion, taking into account potentialities and limitations, the proposed approach can be considered able to support sustainable decision-making, being applicable in other regions.
https://doi.org/10.1590/0001-3765201720160915
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7.
Diretriz de Telecardiologia no Cuidado de Pacientes com Síndrome Coronariana Aguda e Outras Doenças Cardíacas
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Oliveira Junior, Mucio Tavares de
; Canesin, Manoel Fernandes
; Marcolino, Milena Soriano
; Ribeiro, Antonio Luiz Pinho
; Carvalho, Antonio Carlos de Camargo
; Reddy, Shankar
; Santos, Adson Roberto França dos
; Fernandes, Alfredo Manoel da Silva
; Amaral, Amaury Zatorre
; Rezende, Ana Carolina de
; Nechar Junior, Antonio
; Nascimento, Bruno Ramos do
; Pastore, Carlos Alberto
; Wen, Chao Lung
; Gualandro, Danielle Menosi
; Napoli, Domingos Guilherme
; França, Francisco Faustino A. C.
; Feitosa-Filho, Gilson Soares
; Saad, Jamil Abdalla
; Pilli, Jeanne
; Paula, Leonardo Jorge Cordeiro de
; Lodi-Junqueira, Lucas
; Cesar, Luis Antonio Machado
; Bodanese, Luiz Carlos
; Gutierrez, Marco Antonio
; Alkmim, Maria Beatriz Moreira
; Nunes, Mauricio Batista
; Medeiros, Orlando Otávio de
; Moreno, Ramon Alfredo
; Gundim, Rosângela Simões
; Montenegro, Sergio Tavares
; Nazima, Willyan Issamu
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https://doi.org/10.5935/abc.20150057
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8.
Skin impression with acetate tape in Demodex canis and Scarcoptes scabiei var. vulpes diagnosis
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Arquivo Brasileiro de Medicina Veterinária e Zootecnia
- Métricas do periódico
Este estudo compara a eficácia da impressão cutânea com fita de acetato ao raspado cutâneo profundo para a pesquisa de D. canis e S. scabiei. Em um período de seis meses, foram coletadas 134 amostras de cada uma das técnicas de um total de 115 cães atendidos na rotina dermatológica do Hospital Veterinário Universitário da Universidade Federal de Santa Maria (HVU-UFSM). Desses pacientes, 27 cães apresentavam sarna demodécica e 12 cães, escabiose. A impressão cutânea com fita de acetato, quando comparada ao raspado cutâneo profundo, demonstrou ser significativamente superior na pesquisa dos ácaros D. canis e S. scabiei (p = 0,007). Conclui-se que o método da fita de acetato pode ser usado em substituição ao raspado profundo de pele para o diagnóstico e controle da terapia das enfermidades dermatológicas produzidas por ácaros. Além de ser um método sensível, ele é menos traumático para o animal, sendo, dessa forma, mais aceito pelo proprietário.
This study compares the efficacy of skin impression with acetate tape and the deep skin scraping test to find D. canis and S. scabieiin dogs. During six months, 134 samples were collected by both techniques from 115 dogs treated at the dermatology service of the Veterinary Hospital of the Federal University of Santa Maria (HVU-UFSM). Of these patients, 27 had demodicosis and 12 had scabies. The impression with acetate tape test (ITT) was shown to be significantly superior to the deep skin scraping test (DSST) in finding D. canis and S. scabiei mites (p = 0.007). Based on our results we could conclude that acetate tape impression is a reliable method for diagnosing and monitoring therapy of dermatopathies caused by mites and can be used to replace the traditional deep skin scraping method. In addition, since it is less traumatic for the dog, this method shows more acceptance by the owner.
https://doi.org/10.1590/1678-6869
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Growing knowledge: an overview of Seed Plant diversity in Brazil
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Zappi, Daniela C.
; Filardi, Fabiana L. Ranzato
; Leitman, Paula
; Souza, Vinícius C.
; Walter, Bruno M.T.
; Pirani, José R.
; Morim, Marli P.
; Queiroz, Luciano P.
; Cavalcanti, Taciana B.
; Mansano, Vidal F.
; Forzza, Rafaela C.
; Abreu, Maria C.
; Acevedo-Rodríguez, Pedro
; Agra, Maria F.
; Almeida Jr., Eduardo B.
; Almeida, Gracineide S.S.
; Almeida, Rafael F.
; Alves, Flávio M.
; Alves, Marccus
; Alves-Araujo, Anderson
; Amaral, Maria C.E.
; Amorim, André M.
; Amorim, Bruno
; Andrade, Ivanilza M.
; Andreata, Regina H.P.
; Andrino, Caroline O.
; Anunciação, Elisete A.
; Aona, Lidyanne Y.S.
; Aranguren, Yani
; Aranha Filho, João L.M.
; Araújo, Andrea O.
; Araújo, Ariclenes A.M.
; Araújo, Diogo
; Arbo, María M.
; Assis, Leandro
; Assis, Marta C.
; Assunção, Vivian A.
; Athiê-Souza, Sarah M.
; Azevedo, Cecilia O.
; Baitello, João B.
; Barberena, Felipe F.V.A.
; Barbosa, Maria R.V.
; Barros, Fábio
; Barros, Lucas A.V.
; Barros, Michel J.F.
; Baumgratz, José F.A.
; Bernacci, Luis C.
; Berry, Paul E.
; Bigio, Narcísio C.
; Biral, Leonardo
; Bittrich, Volker
; Borges, Rafael A.X.
; Bortoluzzi, Roseli L.C.
; Bove, Cláudia P.
; Bovini, Massimo G.
; Braga, João M.A.
; Braz, Denise M.
; Bringel Jr., João B.A.
; Bruniera, Carla P.
; Buturi, Camila V.
; Cabral, Elza
; Cabral, Fernanda N.
; Caddah, Mayara K.
; Caires, Claudenir S.
; Calazans, Luana S.B.
; Calió, Maria F.
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; Carauta, Jorge P.P.
; Cardiel, José M.
; Cardoso, Domingos B.O.S.
; Cardoso, Leandro J.T.
; Carneiro, Camila R.
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; Carneiro-Torres, Daniela S.
; Carrijo, Tatiana T.
; Caruzo, Maria B.R.
; Carvalho, Maria L.S.
; Carvalho-Silva, Micheline
; Castello, Ana C.D.
; Cavalheiro, Larissa
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; Chacon, Roberta G.
; Chautems, Alain
; Chiavegatto, Berenice
; Chukr, Nádia S.
; Coelho, Alexa A.O.P.
; Coelho, Marcus A.N.
; Coelho, Rubens L.G.
; Cordeiro, Inês
; Cordula, Elizabeth
; Cornejo, Xavier
; Côrtes, Ana L.A.
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; Cota, Maria R.C.
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; Duarte, Marília C.
; Dutilh, Julie H.A.
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; Ferreira, D.M.C.
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; Fiaschi, Pedro
; Filgueiras, Tarciso S.
; Firens, Marcela
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; França, Flávio
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; Gonçalves, Eduardo Gomes
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; Guimarães, Elsie F.
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; Harley, Raymond
; Hassemer, Gustavo
; Hattori, Eric K.O.
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; Henderson, Andrew
; Hensold, Nancy
; Hiepko, Paul
; Holanda, Ana S.S.
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; Indriunas, Alexandre
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; Jardim, Jomar G.
; Kamer, Hiltje M.
; Kameyama, Cíntia
; Kinoshita, Luiza S.
; Kirizawa, Mizué
; Klitgaard, Bente B.
; Koch, Ingrid
; Koschnitzke, Cristiana
; Krauss, Nathália P.
; Kriebel, Ricardo
; Kuntz, Juliana
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; Leal, Eduardo S.
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; Lima, Itamar B.
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; Lima, Rita B.
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; Lombardi, Julio A.
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; Medeiros, João D.
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; Monteiro, Daniele
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; Mota, Nara F.O.
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; Mulgura, Maria
; Nakajima, Jimi N.
; Nardy, Camila
; Nascimento Júnior, José E.
; Noblick, Larry
; Nunes, Teonildes S.
; O'Leary, Nataly
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; Oliveira, Caetano T.
; Oliveira, Juliana A.
; Oliveira, Luciana S.D.
; Oliveira, Maria L.A.A.
; Oliveira, Regina C.
; Oliveira, Renata S.
; Oliveira, Reyjane P.
; Paixão-Souza, Bruno
; Parra, Lara R.
; Pasini, Eduardo
; Pastore, José F.B.
; Pastore, Mayara
; Paula-Souza, Juliana
; Pederneiras, Leandro C.
; Peixoto, Ariane L.
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; Pellegrini, Marco O.O.
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; Perdiz, Ricardo O.
; Pereira, Anna C.M.
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; Pessoa, Clenia
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; Proença, Carolyn
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; Queiroz, George A.
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; Ritter, Mara R.
; Rivadavia, Fernando
; Rocha, Antônio E.S.
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; Rodrigues, Karina F.
; Rodrigues, Rodrigo S.
; Rodrigues, Rodrigo S.
; Rodrigues, Vinícius T.
; Rodrigues, William
; Romaniuc Neto, Sérgio
; Romão, Gerson O.
; Romero, Rosana
; Roque, Nádia
; Rosa, Patrícia
; Rossi, Lúcia
; Sá, Cyl F.C.
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; Saka, Mariana
; Sakuragui, Cássia M.
; Salas, Roberto M.
; Sales, Margareth F.
; Salimena, Fatima R.G.
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; Sancho, Gisela
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; Scalon, Viviane R.
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; Sebastiani, Renata
; Secco, Ricardo S.
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; Senna-Valle, Luci
; Shirasuna, Regina T.
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; Silva, Márcia C.R.
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; Silva, Saura R.
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; Silva-Gonçalves, Kelly C.
; Silva-Luz, Cíntia L.
; Simão-Bianchini, Rosângela
; Simões, André O.
; Simpson, Beryl
; Siniscalchi, Carolina M.
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; Siqueira, Josafá C.
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; Snak, Cristiane
; Soares Neto, Raimundo L.
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; Sobral, Marcos
; Sodré, Rodolfo C.
; Somner, Genise V.
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; Sousa, Danilo J.L.
; Souza, Elnatan B.
; Souza, Élvia R.
; Souza, Marcelo
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Resumo Um levantamento atualizado das plantas com sementes e análises relevantes acerca desta biodiversidade são apresentados. Este trabalho se iniciou em 2010 com a publicação do Catálogo de Plantas e Fungos e, desde então vem sendo atualizado por mais de 430 especialistas trabalhando online. O Brasil abriga atualmente 32.086 espécies nativas de Angiospermas e 23 espécies nativas de Gimnospermas e estes novos dados mostram um aumento de 3% da riqueza em relação a 2010. A Amazônia é o Domínio Fitogeográfico com o maior número de espécies de Gimnospermas, enquanto que a Floresta Atlântica possui a maior riqueza de Angiospermas. Houve um crescimento considerável no número de espécies e nas taxas de endemismo para a maioria dos Domínios (Caatinga, Cerrado, Floresta Atlântica, Pampa e Pantanal), com exceção da Amazônia que apresentou uma diminuição de 2,5% de endemicidade. Entretanto, a maior parte das plantas com sementes que ocorrem no Brasil (57,4%) é endêmica deste território. A proporção de formas de vida varia de acordo com os diferentes Domínios: árvores são mais expressivas na Amazônia e Floresta Atlântica do que nos outros biomas, ervas são dominantes no Pampa e as lianas apresentam riqueza expressiva na Amazônia, Floresta Atlântica e Pantanal. Este trabalho não só quantifica a biodiversidade brasileira, mas também indica as lacunas de conhecimento e o desafio a ser enfrentado para a conservação desta flora.
Abstract An updated inventory of Brazilian seed plants is presented and offers important insights into the country's biodiversity. This work started in 2010, with the publication of the Plants and Fungi Catalogue, and has been updated since by more than 430 specialists working online. Brazil is home to 32,086 native Angiosperms and 23 native Gymnosperms, showing an increase of 3% in its species richness in relation to 2010. The Amazon Rainforest is the richest Brazilian biome for Gymnosperms, while the Atlantic Rainforest is the richest one for Angiosperms. There was a considerable increment in the number of species and endemism rates for biomes, except for the Amazon that showed a decrease of 2.5% of recorded endemics. However, well over half of Brazillian seed plant species (57.4%) is endemic to this territory. The proportion of life-forms varies among different biomes: trees are more expressive in the Amazon and Atlantic Rainforest biomes while herbs predominate in the Pampa, and lianas are more expressive in the Amazon, Atlantic Rainforest, and Pantanal. This compilation serves not only to quantify Brazilian biodiversity, but also to highlight areas where there information is lacking and to provide a framework for the challenge faced in conserving Brazil's unique and diverse flora.
https://doi.org/10.1590/2175-7860201566411
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10.
Plant species used in giardiasis treatment: ethnopharmacology and in vitro evaluation of anti-Giardia activity
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Neiva, Vanessa do A.
; Ribeiro, Maria Nilce S.
; Nascimento, Flávia R. F.
; Cartágenes, Maria do Socorro S.
; Coutinho-Moraes, Denise F.
; Amaral, Flavia M. M. do
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Revista Brasileira de Farmacognosia
- Métricas do periódico
The aim of this study was to compile the traditional knowledge about plants used for the treatment of giardiasis, and also to carry out experimental research to evaluate the anti-Giardia activity of five species.To reach this objective, 398 interviews were performed using a previously prepared questionnaire, followed by an in vitro evaluation of giardicidal potential of hydroalcoholic leaf extracts of Anacardium occidentale L., Chenopodium ambrosioides L., Passiflora edulis Sims, Psidium guajava L., and Stachytarpheta cayennensis(Rich.) Vahl. Among the interviewed people, 55.53% reported the use of plants to treat diarrhea, the most severe symptom of giardiasis. The results indicated 36 species used by this population for these problems. The use of leaves (72.50%) of a single plant (64.25%) collected from backyards and gardens (44.34%) and prepared by decoction were predominant. The majority of the interviewees (85.52%) attributed their cure to the use of plants. In the experimental tests, all extracts inhibited the growth of Giardia lambliatrophozoites in different intensities: A. occidentale and P. guajava extracts elicited a moderate activity (250 ≤ IC50 ≤ 500 μg/ml), C. ambrosioides and S. cayennensis extracts evoked a high activity (100 ≤ IC50 ≤ 250 μg/ml), and P. edulis extract showed very high activity (IC50≤ 100 μg/ml). This study shows that an ethnopharmacological approach is useful in the selection of plant materials with potential giardicidal activity.
https://doi.org/10.1016/j.bjp.2014.04.004
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11.
Mutação G20210A no gene da protrombina, fator V de Leiden e anticorpos anticardiolipina não influenciam a sobrevida do enxerto renal após o transplante
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Rocha, Luis Klaus A. da
; Galante, Nelson Zocoler
; Alvarez, Vivian Angélica Castilho
; Areco, Kelsy C. N.
; Noguti, Maria Aparecida E.
; Amaral, Rogério Q.
; Andrade, Luis Eduardo C.
; Peres, Clóvis Araujo
; Pestana, José O. Medina
; Lourenço, Dayse M.
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INTRODUÇÃO: Complicações tromboembólicas são importantes fatores de risco para perda do enxerto e pior evolução após o transplante renal. Pacientes com defeito trombofílico apresentam maior risco de complicações tromboembólicas. Foram analisados, entre receptores de transplante renal, a prevalência de defeito trombofílico e o risco atribuído a esta condição para a perda do enxerto e para o desenvolvimento de tromboses intravasculares. MÉTODOS: Estudo do tipo coorte incluindo 388 receptores adultos analisados quanto à presença de trombofilia de acordo com a pesquisa de anticorpos anticardiolipina (aCL) por ELISA e das mutações G1691A no gene do fator V (FV) e G20210A no gene da protrombina (PT) por PCR multiplex. RESULTADOS: Defeito trombofílico foi identificado em 25,8% dos pacientes. As taxas de sobrevida de 2 anos do enxerto foram semelhantes entre os pacientes com e sem defeito trombofílico (94% versus 94%, p = 0,53), bem como a sobrevida dos enxertos livres de tromboses intravasculares (97% versus 97%, p = 0,83). Pacientes com defeito trombofílico apresentaram prevalência de tromboses intravasculares semelhante à do grupo-controle (3% versus 3,5%, p = 0,82). O transplante renal anterior foi associado a maior risco de perda de enxerto (OR 20,8, p < 0,001) e de ocorrência de tromboses intravasculares (OR 6,8, p = 0,008). CONCLUSÕES: As prevalências das mutações FV G1691A e PT G20210A na população estudada foram semelhantes às da população geral não transplantada, e a prevalência de anticorpos aCL superou a observada entre os indivíduos sadios. Não houve associação entre os marcadores de trombofilia estudados e a sobrevida em médio prazo do transplante renal.
INTRODUCTION: Thromboembolic complications are important risk factors for graft failure and worse renal transplantation outcome. Patients with thrombophilic disorders have a higher risk of thromboembolic complications. The prevalence of thrombophilic disorders and the associated risk for graft failure and for intravascular thrombosis were analyzed in renal transplant recipients. METHODS: This is a cohort study of 388 adult recipients investigated regarding the presence of thrombophilia, through the search for anticardiolipin antibodies (aCL) via ELISA and FV G1691A and PT G20210A gene mutations by multiplex PCR. RESULTS: Thrombophilic disorders were identified in 25.8% of the patients. The 2-year graft survival was similar among patients with and without thrombophilic disorder (94% versus 94%, p = 0.53), and so was the survival free of intravascular thrombosis (97% versus 97%, p = 0.83). The prevalence of intravascular thrombosis was similar in both groups (3% versus 3.5%, p = 0.82). Patients with previous kidney transplantation had a higher risk of graft failure (OR 20.8, p < 0.001) and of intravascular thrombosis (OR 6.8, p = 0.008). CONCLUSIONS: The prevalences of FV G1691A and PT G20210A gene mutations in this cohort of patients were similar to those of the general non-transplanted population. The prevalence of aCL antibodies was higher in this cohort than that observed in healthy individuals. The thrombophilic markers studied did not predict the medium-term survival of renal transplant.
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12.
Influência do subsídio financeiro e do local da realização do curso de suporte avançado de vida em cardiologia, no aprendizado da emergência cardiovascular
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Miotto, Heberth C.
; Goulart, Eugênio M. A.
; Amaral, Carlos Faria Santos
; Moreira, Maria da Consolação V.
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Arquivos Brasileiros de Cardiologia
- Métricas do periódico
FUNDAMENTO: O sucesso no aprendizado da emergência depende de muitos fatores que podem ser resumidos como: aluno, instrutores e curso. OBJETIVO: Avaliar a influência do subsídio financeiro e do local da realização do curso no aprendizado da emergência cardiovascular. MÉTODOS: Analisaram-se dados referentes aos cursos de Suporte Avançado de Vida em Cardiologia (ACLS) no período de dezembro de 2005 a dezembro de 2006. De acordo com o subsídio financeiro, foram divididos em: grupo 1 - subsídio integral; grupo 2 - subsídio de 50%; e grupo 3 - sem subsídio. Quanto ao local do curso, foram divididos em: local A - curso em cidade com > 1 milhão de habitantes; e local B - curso em cidade com < 1 milhão de habitantes. Compararam-se a aprovação prática e teórica e a média teórica. RESULTADOS: Participaram do ACLS 819 alunos: 199 (24%) no grupo 1, 122 (15%) no 2 e 498 (61%) no 3. A aprovação prática e teórica e a média na prova teórica foram maiores no grupo 3 que nos demais grupos (p<0,05). Quatrocentos e oitenta e dois fizeram o curso no local A (59%) e 337 (41%) no local B. A aprovação prática foi semelhante para ambos os grupos (p = 0,33), entretanto a aprovação teórica foi maior no local A (73% vs. 65% - p = 0,021 - OR = 1,44 e IC: 1,05 - 1,97). A média teórica foi maior no local A (87,1 ± 10,4 e 86 ± 11, respectivamente p<0,05). CONCLUSÃO: O subsídio financeiro e o local da realização do curso influenciaram na aprovação teórica e prática.
BACKGROUND: The success in learning of emergency depends on many factors that can be summarized as: student, instructors and course. OBJECTIVE: To evaluate the influence of financial subsidy and venue of course in learning cardiovascular emergency. METHODS: Data were analyzed regarding the courses of Advanced Cardiac Life Support (ACLS) in the period from December 2005 to December 2006. In agreement with the financial subsidy, they were divided in: group 1 - integral subsidy; group 2 - subsidy of 50%; and group 3 - without subsidy. As for the venue of the course, they were divided in: locality A - study in city with> 1 million inhabitants; and locality B - study in city with <1 million inhabitants. The practical and theoretical approval and the theoretical average were compared. RESULTS: 819 students participated in ACLS: 199 (24%) in group 1, 122 (15%) in 2 and 498 (61%) in 3. The practical and theoretical approval and the average in the theoretical exam were greater in group 3 than in other groups (p <0.05). Four hundred and eighty two (482) took the course in venue A (59%) and 337 (41%) in venue B. The practical approval was similar for both groups (p = 0.33), however the theoretical approval was greater in venue A (73% vs. 65% - p = 0.021 - OR = 1.44 and IC: 1.05 - 1.97). The theoretical average was greater in venue A (87.1 ± 10.4 and 86 ± 11, respectively p <0.05). CONCLUSION: The financial subsidy and venue of the course had influence in the theoretical and practical approval.
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13.
Feeding and oviposition preference of Phyllophaga cuyabana (Moser) (Coleoptera: Melolonthidae) on several crops
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Estudos em laboratório e em casa-de-vegetação foram conduzidos para estudar a preferência de Phyllophaga cuyabana (Moser) em se alimentar e ovipositar nas espécies de plantas: Cajanus cajan L. (guandu), Crotalaria juncea L. (crotalária), Crotalaria spectabilis Roth (crotalária), Crotalaria ochroleuca G. Don (crotalária), Glycine max [L.] Merrill (soja), Gossypium hirsutum L. (algodão), Helianthus annuus L. (girassol), Stizolobium aterrimum [Mucuna aterrima] Piper & Tracey (mucuna preta) e Zea mays L. (milho). O maior número de ovos foi observado em girassol, C. juncea e soja e o menor em algodão, em situação de confinamento. Em testes de multipla-escolha, os adultos não fizeram discriminação entre as plantas. Entretanto, em teste de dupla-escolha, a proporção de ovos e do consumo foliar em soja foi significativamente maior do que em C. spectabilis. Em situação de múltipla escolha, a distribuição das larvas ocorreu ao acaso, não sendo observada nenhuma tendência de preferência, mas em situação de dupla-escolha, usando-se soja como padrão, as larvas sempre preferiram se alimentar nas raízes de soja. Os adultos de P. cuyabana preferiram os hospedeiros mais adequados à sobrevivência de sua prole. Esse comportamento pode ser explorado em um programa de manejo integrado dessa praga.
Laboratory and greenhouse experiments were carried out to study food and oviposition preference by Phyllophaga cuyabana (Moser) on different plant species as Cajanus cajan L. (pigeon pea), Crotalaria juncea L. (sun hemp), Crotalaria spectabilis Roth (showy crotalaria), Crotalaria ochroleuca G. Don (slenderleaf rattlebox), Glycine max [L.] Merrill (soybean), Gossypium hirsutum L. (cotton), Helianthus annuus L. (sunflower), Stizolobium aterrimum [Mucuna aterrima] Piper & Tracey (velvetbean) and Zea mays L. (mayze). In no-choice experiments, the number of eggs layed in sunflower, C. juncea and soybean was larger compared to cotton. Despite the fact that the adults did not discriminate among plants, in dual-choice test, the proportion of eggs layed and leaf consumption by P. cuyabana adults in soybean were significantly higher than in C. spectabilis. The larval distribution in the soil was at random in multiple-choice, withouth any trend of preference, but in dual-choice, when soybean was the control, larvae always preferred to feed on its roots. P. cuyabana adults had preference for more suitable hosts and that could stand their offspring survival. This behaviour can be usefully exploited in an integrated management program for this pest.
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14.
Abietane diterpenes from Sagittaria montevidensis ssp montevidensis Charm. & Schltdl
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Radke, Vanessa S. C. de O.
; Amaral, Maria do Carmo E.
; Schuquel, Ivânia T. A.
; Silva, Cleuza C. da
; Oliveira, Cecília M. A. de
; Tanaka, Clara M. A.
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Journal of the Brazilian Chemical Society
- Métricas do periódico
Dois novos diterpenos do tipo abietano 3beta-hidroxi-9alfa, 13alfa-epidioxiabiet-8(14)-eno (1) e 3-oxo-9alfa,13alfa-epidioxiabiet-8(14)-eno (2) foram isolados do extrato bruto metanólico dos pecíolos de Sagittaria montevidensis ssp montevidensis (Alismataceae). As estruturas de 1 e 2 foram determinadas com base em análises espectrométricas do tipo EM-AR, IV, bem como, RMN de ¹H e 13C uni e bi dimensionais.
Two new abietane-type diterpenes, 3beta-hydroxy-9alpha, 13alpha-epidioxyabiet-8(14)-ene (1) and 3-oxo-9alpha,13alpha-epidioxyabiet-8(14)-ene (2), were isolated from the methanolic crude extract of the petioles of Sagittaria montevidensis ssp montevidensis (Alismataceae). The structures of 1 and 2 were determined on the basis of spectrometric analyses including HREIMS, IR as well as ¹H and 13C 1 and 2D NMR.
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15.
Analysis of expressed sequence tags from Citrus sinensis L. Osbeck infected with Xylella fastidiosa
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Souza, Alessandra A. de
; Takita, Marco A.
; Coletta-Filho, Helvécio D.
; Targon, Maria Luisa P.N.
; Carlos, Eduardo F.
; Locali-Fabris, Eliane C.
; Amaral, Alexandre M.
; Freitas-Astúa, Juliana
; Silva-Pinhati, Ana Carla O.
; Boscariol-Camargo, Raquel L.
; Berger, Irving J.
; Rodrigues, Carolina M.
; Reis, Marcelo S.
; Machado, Marcos A.
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In order to understand the genetic responses resulting from physiological changes that occur in plants displaying citrus variegated chlorosis (CVC) symptoms, we adopted a strategy of comparing two EST libraries from sweet orange [Citrus sinensis (L.) Osbeck]. One of them was prepared with plants showing typical CVC symptoms caused by Xylella fastidiosa and the other with non-inoculated plants. We obtained 15,944 ESTs by sequencing the two cDNA libraries. Using an in silico hybridization strategy, 37 genes were found to have significant variation at the transcriptional level. Within this subset, 21 were up-regulated and 16 were down-regulated in plants with CVC. The main functional categories of the down-regulated transcripts in plants with CVC were associated with metabolism, protein modification, energy and transport facilitation. The majority of the up-regulated transcripts were associated with metabolism and defense response. Some transcripts associated with adaptation to stress conditions were up-regulated in plants with CVC and could explain why plants remain alive even under severe water and nutritional stress. Others of the up-regulated transcripts are related to defense response suggesting that sweet orange plants activate their defense machinery. The genes associated with stress response might be expressed as part of a secondary response related to physiological alterations caused by the infection.
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