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1.
A rare case of granulomatous slack skin with scarce multinucleated giant cells
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Hollanda, Laísa E. de
; Oliveira, Carolina S. de
; Mendes-Alexandre, Isabella C.
; Alves-Melo-Martins, Rebeca de O.
; Ferreira, Vanessa R.
; Reis, Monique F. dos
; Damasceno-Ferreira, Silvana de A.
; Santos, Luciana M. dos
.
Portuguese Journal of Dermatology and Venereology
- Métricas do periódico
2.
Impact of Conservation Processes on the Lipid Profile and Immunological Factors IL-10 and TGF-β1 in Whey Separated from Discarded Human Milk IL10 IL 10 IL-1 TGFβ1 TGFβ TGF β1 β TGF-β IL1 1 IL-
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Alves, Eloize S.
; Castro, Matheus C.
; Saqueti, Bruno H. F.
; Manin, Luciana P.
; Alencar, Josiane B.
; Zacarias, Joana M. V.
; Bruni, Andressa R. S.
; Madrona, Grasiele S.
; Visentainer, Jeane E. L.
; Cristianini, Marcelo
; Santos, Oscar O.
; Visentainer, Jesui V.
.
Journal of the Brazilian Chemical Society
- Métricas do periódico
Reuse made by the separation of whey can reduce the waste of human milk. However, the authors are not aware of the literature on treatments in human whey, made available by pasteurization holder, freeze-drying, spray drying, and high hydrostatic pressure. In this context, the present study applied treatments to human whey and evaluated their lipid and immunological quality. Among the results, a different formation in the triacylglycerol profile was evidenced after the application of spray drying and high hydrostatic pressure, while pasteurization and freeze-drying presented ion intensity close to the control human whey. In addition, pasteurization proved to be adequate for lipid nutritional quality and transformation factor-β1 (TGF-β1) concentration, while an increase in interleukin-10 (IL-10) levels was promoted, between 73 and 80%, after freeze-drying, spray drying, and high hydrostatic pressure. Through the principal component analysis, it is noteworthy that the processes presented divergences in terms of the effects caused, with similarity only between pasteurization and freeze-drying in the composition of fatty acids. However, it was observed that all processes were able to maintain the nutrients. Nevertheless, it is relevant to consider individual characteristics presented and the interest in the desired quality, which can be promising as a complementary product to infant feeding. milk However holder freezedrying, freezedrying freeze pressure context results addition factorβ1 factorβ factor β1 β factor-β TGFβ1 TGFβ TGF (TGF-β1 concentration interleukin10 interleukin 10 interleukin-1 IL10 IL (IL-10 promoted 7 80 80% analysis caused acids nutrients Nevertheless feeding (TGF-β interleukin1 1 interleukin- IL1 (IL-1 8 (IL- (IL
3.
Lavandula dentata L. essential oil: a promising antifungal and antibiofilm agent against oral Candida albicans L oil
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Santos, A. A.
; Oliveira-Filho, A. A.
; Teixeira, B. A.
; Borchardt, H.
; Galvão, J. L. F. M.
; Medeiros, M. A. A.
; Alves, M. S.
; Barbosa, D. H. X.
; Mafra, R. P.
; Nascimento, Y. M.
; Vasconcelos, U.
; Lima, E. O.
.
Abstract Candida albicans is the main fungal species involved in oral candidiasis, and its increasing resistance to pharmacological treatment encourages the search for improved antifungal agents. Lavandula dentata L. essential oil (LD-EO) has been recognized for its antimicrobial activity, but little is known about its role against oral C. albicans. This study evaluated the antifungal and antibiofilm activities, mechanisms of action, and toxicity of LD-EO from Brazil against oral strains of C. albicans. Antifungal activity was assessed based on Minimum Inhibitory Concentration (MIC), Minimum Fungicidal Concentration (MFC), association study with miconazole (Checkerboard method), and sorbitol and ergosterol assays. Inhibition of biofilm formation and disruption of preformed biofilm were considered when studying the effects of the product. Additionally, the toxicity of LD-EO was evaluated by a hemolysis assay on human erythrocytes. Phytochemical analysis by gas chromatography-mass spectrometry identified eucalyptol (33.1%), camphor (18.3%), and fenchone (15.6%) as major constituents. The test substance showed mainly fungicidal activity (MIC100 = 8 μg/mL; MFC = 16 μg/mL), including against two miconazole-resistant isolates of C. albicans. The effects of LD-EO were synergistic with those of miconazole and appeared not to involve damage to the fungal cell wall or plasma membrane. Its effectiveness in inhibiting biofilm formation was higher than the effect of disrupting preformed biofilm. Finally, the product exhibited low hemolytic activity at MIC. Based on the favorable and novel results described here, LD-EO could constitute a promising therapeutic alternative for oral candidiasis, including miconazole-resistant cases. candidiasis agents L LDEO LD EO (LD-EO C activities action MIC, MIC , (MIC) MFC, (MFC) Checkerboard method, method method) assays Additionally erythrocytes chromatographymass chromatography mass 33.1%, 331 33.1% 33 1 (33.1%) 18.3%, 183 18.3% 18 3 (18.3%) 15.6% 156 15 6 (15.6% constituents MIC100 (MIC10 μg/mL μgmL μg mL μg/mL, μg/mL) miconazoleresistant resistant membrane Finally here cases (MIC (MFC 33.1 (33.1% 18.3 (18.3% 15.6 (15.6 MIC10 (MIC1 33. (33.1 18. (18.3 15. (15. MIC1 (33. (18. (15 (33 (18 (1 (3 (
Resumo Candida albicans é a principal espécie fúngica envolvida na candidíase bucal, e sua crescente resistência ao tratamento farmacológico encoraja a busca por melhores agentes antifúngicos. O óleo essencial da Lavandula dentata L. (LD-EO) tem sido reconhecido por sua atividade antimicrobiana, porém pouco se conhece o seu papel contra C. albicans bucal. Este trabalho avaliou as atividades antifúngica e antibiofilme, mecanismos de ação e toxicidade do LD-EO do Brasil contra cepas de C. albicans bucal. A atividade antifúngica foi avaliada baseando-se em: Concentração Inibitória Mínima (CIM), Concentração Fungicida Mínima (CFM), estudo de associação com o miconazol (método Checkerboard) e ensaios com sorbitol e ergosterol. A inibição da formação do biofilme e a ruptura do biofilme pré-formado foram considerados no estudo dos efeitos do produto. Adicionalmente, a toxicidade do LD-EO foi avaliada pelo ensaio de hemólise em eritrócitos humanos. A análise fitoquímica por cromatografia gasosa-espectrometria de massa identificou eucaliptol (33.1%), cânfora (18.3%) e fenchona (15.6%) como constituintes majoritários. A substância teste revelou atividade principalmente fungicida (CIM100 = 8 μg/mL; CFM = 16 μg/mL), inclusive contra dois isolados de C. albicans resistentes ao miconazol. Os efeitos do LD-EO foram sinérgicos aos do miconazol e parecem não envolver danos à parede celular ou à membrana plasmática fúngica. Sua efetividade em inibir a formação do biofilme foi maior que o efeito de eliminação do biofilme pré-formado. Finalmente, o produto exerceu baixa atividade hemolítica na CIM. Considerando os resultados favoráveis e inéditos aqui descritos, o LD-EO poderia constituir uma alternativa terapêutica promissora para a candidíase bucal, incluindo casos resistentes ao miconazol. bucal antifúngicos L LDEO LD EO (LD-EO antimicrobiana C antibiofilme baseandose baseando CIM, CIM , (CIM) CFM, (CFM) método Checkerboard ergosterol préformado pré formado Adicionalmente humanos gasosaespectrometria gasosa espectrometria 33.1%, 331 33.1% 33 1 (33.1%) 18.3% 183 18 3 (18.3% 15.6% 156 15 6 (15.6% majoritários CIM100 (CIM10 μg/mL μgmL μg mL μg/mL, μg/mL) préformado. formado. Finalmente descritos (CIM (CFM 33.1 (33.1% 18.3 (18.3 15.6 (15.6 CIM10 (CIM1 33. (33.1 18. (18. 15. (15. CIM1 (33. (18 (15 (33 (1 (3 (
4.
Biometric aspects of fruits and seeds and determination of the absorption curve of Hymenaea martiana Hayne seeds
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Silva, M. J.
; Alves, E. U.
; Silva, J. N.
; Silva, R. S.
; Bernardo, M. K. F.
; Rodrigues, C. M.
; Pádua, G. V. G.
; Silva, J. H. C. S.
; Silva, M. C. L.
; Souza, A. G.
; Smiderle, O. J.
.
Abstract The biometric differences between fruits and seeds are useful characteristics that can provide important data for the investigation and preservation of the species and may be linked to environmental and genetic influences. In this sense, considering the importance of this species and the need for conservation, the objective was to carry out physical characterization of the fruits and seeds of Hymenaea martiana as well as to determine the seed imbibition curve. The experiment was conducted at the Seed Analysis Laboratory at the Agricultural Sciences Center at the Federal University of Paraíba in Areia, PB. The evaluations carried out were as follows: biometry of fruits and seeds, number of seeds per fruit, colorimetry of fruits and seeds, percentage of damaged seeds, weight of a thousand seeds, seed water content, mass and imbibition curve. The biometric data were subjected to descriptive analysis to determine the minimum, maximum, average value, standard deviation, asymmetry, and kurtosis of the fruits and seeds. In terms of the biometric characteristics of the fruits and seeds of H. martiana, there was a marked variation, with average fruit lengths of 90.28 mm, widths of 46.83 mm, thicknesses of 34.69 mm, weights of 65.86 g and four seeds per fruit. The average length, width, thickness and weight of the seeds were 23.75 mm, 18.34 mm, 12.71 g and 4.13 g, respectively. The fruits were darker than the seeds, and both the fruits and seeds had red tones. Compared with nonscarified seeds, scarified seeds absorb a greater amount of water. influences sense conservation curve Areia PB follows content minimum maximum value deviation asymmetry H variation 9028 90 28 90.2 mm 4683 46 83 46.8 3469 34 69 34.6 6586 65 86 65.8 length width 2375 23 75 23.7 1834 18 18.3 1271 12 71 12.7 413 4 13 4.1 respectively tones 902 9 2 90. 468 8 46. 346 3 6 34. 658 65. 237 7 23. 183 1 18. 127 12. 41 4.
Resumo As diferenças biométricas entre frutos e sementes são características úteis que podem fornecer dados importantes para a investigação e preservação da espécie, podendo estar vinculadas a influências ambientais e genéticas. Neste sentido, considerando a importância dessa espécie e a necessidade de conservação, objetivou-se realizar a caracterização física dos frutos e sementes de Hymenaea martiana, bem como determinar a curva de embebição das sementes. O experimento foi conduzido no Laboratório de Análise de Sementes, do Centro de Ciências Agrárias, da Universidade Federal da Paraíba, em Areia - PB. As avaliações realizadas foram as seguintes: biometria de frutos e sementes, número de sementes por frutos, colorimetria dos frutos e sementes, porcentagem de sementes danificadas, peso de mil sementes, teor de água das sementes, massa e curva de embebição. Os dados biométricos foram submetidos à análise descritiva para determinação do valor mínimo, máximo, médio, desvio padrão, assimetria, curtose dos frutos e sementes. Nas características biométricas de frutos e sementes de H. martiana houve variação acentuada, cujos valores médios dos frutos foram de 90,28 mm para o comprimento, 46,83 mm de largura, 34,69 de espessura, peso de 65,86 g e quatro sementes por fruto. Quanto as sementes, os valores médios foram de 23,75 mm, 18,34 mm, 12,71 e 4,13 g para o comprimento, largura, espessura e peso, respectivamente. Em relação a coloração, foi observado que os frutos são mais escuros que as sementes, e que tanto os frutos quanto as sementes têm tonalidades voltadas para o vermelho. As sementes escarificadas absorvem maior quantidade de água se comparadas as sementes não escarificadas. genéticas sentido conservação objetivouse objetivou Sementes Agrárias Paraíba PB seguintes danificadas mínimo máximo médio padrão assimetria H acentuada 9028 90 28 90,2 comprimento 4683 46 83 46,8 largura 3469 34 69 34,6 6586 65 86 65,8 fruto 2375 23 75 23,7 1834 18 18,3 1271 12 71 12,7 413 4 13 4,1 respectivamente coloração vermelho 902 9 2 90, 468 8 46, 346 3 6 34, 658 65, 237 7 23, 183 1 18, 127 12, 41 4,
5.
Evaluation of miRNAs regulation of BDNF and IGF1 genes in T2DM insulin resistance in experimental models: bioinformatics based approach
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Freitas, R. M.
; Felipe, S. M. S.
; Ribeiro, J. K. C.
; Araújo, V. R.
; Martin, C. P. S.
; Oliveira, M. A. F.
; Martins, S. D.
; Pontes, J. P. A.
; Alves, J. O.
; Soares, P. M.
; Ceccatto, V. M.
.
Resumo Os microRNAs (miRNAs) são reconhecidos como biomarcadores do diabetes mellitus tipo 2 (DM2), úteis para a compreensão do metabolismo da doença, e possuem grande potencial como alvos terapêuticos. O aumento da expressão de BDNF e IGF1 está altamente envolvido nos benefícios as vias de insulina e glicose, porém, são regulados negativamente em condições de resistência à insulina, enquanto seu aumento de expressão está correlacionado com a melhora do metabolismo da glicose e da insulina. Estudos sugerem a regulação desses genes por microRNA em vários contextos diferentes, proporcionando uma nova abordagem de investigação para compreender o metabolismo do DM2 e revelar potenciais alvos terapêuticos. No presente estudo, investigamos em diferentes modelos animais (humanos, ratos e camundongos) miRNAs que têm como alvo BDNF e IGF1 em tecido muscular esquelético com condições fisiológicas de DM2. As análises foram realizadas utilizando ferramentas de bioinformática e bancos de dados para predição de miRNA, homologia molecular, validação experimental de interações, expressão na condição fisiológica estudada e interação em rede. Os resultados mostraram três candidatos a miRNAs para IGF1 (miR-29a, miR-29b e miR-29c) e um para BDNF (miR-206). As avaliações experimentais e a busca pela expressão no músculo esquelético de indivíduos com DM2 confirmaram a interação prevista entre miRNA-mRNA para miR-29b e miR-206 através de modelos humanos, ratos e camundongos. Essa interação foi reafirmada em múltiplas análises de rede. Em conclusão, nossos resultados mostram a relação de regulação entre miR-29b e miR-206 com os genes investigados, em diversos tecidos, sugerindo um padrão de inibição. Contudo, esses dados mostram um grande número de possíveis processos fisiológicos de interação para perspectivas biotecnológicas.
Abstract microRNAs (miRNAs) are recognized as diabetes mellitus type 2 (T2DM) biomarkers useful for disease metabolism comprehension and have great potential as therapeutics targets. BDNF and IGF1 increased expression are highly involved in the benefits of insulin and glucose paths, however, they are down-regulated in insulin resistance conditions, while their expression increase is correlated to the improvement of glucose and insulin metabolism. Studies suggest the microRNA regulation of these genes in several different contexts, providing a novel investigation approach for comprehending T2DM metabolism and revealing potential therapeutic targets. In the present study, we investigate in different animal models (human, rat, and mouse) miRNAs that target BDNF and IGF1 in skeletal muscle tissue with T2DM physiological conditions. Bioinformatics tools and databases were used to miRNA prediction, molecular homology, experimental validation of interactions, expression in the studied physiological condition, and network interaction. The findings showed three miRNAs candidates for IGF1(miR-29a, miR-29b, and miR-29c) and one for BDNF (miR-206). The experimental evaluations and the search for the expression in skeletal muscle from T2DM subjects confirmed the predicted interaction between miRNA-mRNA for miR-29b and miR-206 through human, rat, and mouse models. This interaction was reaffirmed in multiple network analyses. In conclusion, our results show the regulation relationship between miR-29b and miR-206 with the investigated genes, in several tissues, suggesting an inhibition pattern. Nevertheless, these data show a large number of possible interaction physiological processes, for future biotechnological prospects.
6.
Catálogo Taxonômico da Fauna do Brasil: Setting the baseline knowledge on the animal diversity in Brazil Brasil
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Boeger, Walter A.
; Valim, Michel P.
; Zaher, Hussam
; Rafael, José A.
; Forzza, Rafaela C.
; Percequillo, Alexandre R.
; Serejo, Cristiana S.
; Garraffoni, André R.S.
; Santos, Adalberto J.
; Slipinski, Adam
; Linzmeier, Adelita M.
; Calor, Adolfo R.
; Garda, Adrian A.
; Kury, Adriano B.
; Fernandes, Agatha C.S.
; Agudo-Padrón, Aisur I.
; Akama, Alberto
; Silva Neto, Alberto M. da
; Burbano, Alejandro L.
; Menezes, Aleksandra
; Pereira-Colavite, Alessandre
; Anichtchenko, Alexander
; Lees, Alexander C.
; Bezerra, Alexandra M.R.
; Domahovski, Alexandre C.
; Pimenta, Alexandre D.
; Aleixo, Alexandre L.P.
; Marceniuk, Alexandre P.
; Paula, Alexandre S. de
; Somavilla, Alexandre
; Specht, Alexandre
; Camargo, Alexssandro
; Newton, Alfred F.
; Silva, Aline A.S. da
; Santos, Aline B. dos
; Tassi, Aline D.
; Aragão, Allan C.
; Santos, Allan P.M.
; Migotto, Alvaro E.
; Mendes, Amanda C.
; Cunha, Amanda
; Chagas Júnior, Amazonas
; Sousa, Ana A.T. de
; Pavan, Ana C.
; Almeida, Ana C.S.
; Peronti, Ana L.B.G.
; Henriques-Oliveira, Ana L.
; Prudente, Ana L.
; Tourinho, Ana L.
; Pes, Ana M.O.
; Carmignotto, Ana P.
; Wengrat, Ana P.G. da Silva
; Dornellas, Ana P.S.
; Molin, Anamaria Dal
; Puker, Anderson
; Morandini, André C.
; Ferreira, André da S.
; Martins, André L.
; Esteves, André M.
; Fernandes, André S.
; Roza, André S.
; Köhler, Andreas
; Paladini, Andressa
; Andrade, Andrey J. de
; Pinto, Ângelo P.
; Salles, Anna C. de A.
; Gondim, Anne I.
; Amaral, Antonia C.Z.
; Rondón, Antonio A.A.
; Brescovit, Antonio
; Lofego, Antônio C.
; Marques, Antonio C.
; Macedo, Antonio
; Andriolo, Artur
; Henriques, Augusto L.
; Ferreira Júnior, Augusto L.
; Lima, Aurino F. de
; Barros, Ávyla R. de A.
; Brito, Ayrton do R.
; Romera, Bárbara L.V.
; Vasconcelos, Beatriz M.C. de
; Frable, Benjamin W.
; Santos, Bernardo F.
; Ferraz, Bernardo R.
; Rosa, Brunno B.
; Sampaio, Brunno H.L.
; Bellini, Bruno C.
; Clarkson, Bruno
; Oliveira, Bruno G. de
; Corrêa, Caio C.D.
; Martins, Caleb C.
; Castro-Guedes, Camila F. de
; Souto, Camilla
; Bicho, Carla de L.
; Cunha, Carlo M.
; Barboza, Carlos A. de M.
; Lucena, Carlos A.S. de
; Barreto, Carlos
; Santana, Carlos D.C.M. de
; Agne, Carlos E.Q.
; Mielke, Carlos G.C.
; Caetano, Carlos H.S.
; Flechtmann, Carlos H.W.
; Lamas, Carlos J.E.
; Rocha, Carlos
; Mascarenhas, Carolina S.
; Margaría, Cecilia B.
; Waichert, Cecilia
; Digiani, Celina
; Haddad, Célio F.B.
; Azevedo, Celso O.
; Benetti, Cesar J.
; Santos, Charles M.D. dos
; Bartlett, Charles R.
; Bonvicino, Cibele
; Ribeiro-Costa, Cibele S.
; Santos, Cinthya S.G.
; Justino, Cíntia E.L.
; Canedo, Clarissa
; Bonecker, Claudia C.
; Santos, Cláudia P.
; Carvalho, Claudio J.B. de
; Gonçalves, Clayton C.
; Galvão, Cleber
; Costa, Cleide
; Oliveira, Cléo D.C. de
; Schwertner, Cristiano F.
; Andrade, Cristiano L.
; Pereira, Cristiano M.
; Sampaio, Cristiano
; Dias, Cristina de O.
; Lucena, Daercio A. de A.
; Manfio, Daiara
; Amorim, Dalton de S.
; Queiroz, Dalva L. de
; Queiroz, Dalva L. de
; Colpani, Daniara
; Abbate, Daniel
; Aquino, Daniel A.
; Burckhardt, Daniel
; Cavallari, Daniel C.
; Prado, Daniel de C. Schelesky
; Praciano, Daniel L.
; Basílio, Daniel S.
; Bená, Daniela de C.
; Toledo, Daniela G.P. de
; Takiya, Daniela M.
; Fernandes, Daniell R.R.
; Ament, Danilo C.
; Cordeiro, Danilo P.
; Silva, Darliane E.
; Pollock, Darren A.
; Muniz, David B.
; Gibson, David I.
; Nogueira, David S.
; Marques, Dayse W.A.
; Lucatelli, Débora
; Garcia, Deivys M.A.
; Baêta, Délio
; Ferreira, Denise N.M.
; Rueda-Ramírez, Diana
; Fachin, Diego A.
; Souza, Diego de S.
; Rodrigues, Diego F.
; Pádua, Diego G. de
; Barbosa, Diego N.
; Dolibaina, Diego R.
; Amaral, Diogo C.
; Chandler, Donald S.
; Maccagnan, Douglas H.B.
; Caron, Edilson
; Carvalho, Edrielly
; Adriano, Edson A.
; Abreu Júnior, Edson F. de
; Pereira, Edson H.L.
; Viegas, Eduarda F.G.
; Carneiro, Eduardo
; Colley, Eduardo
; Eizirik, Eduardo
; Santos, Eduardo F. dos
; Shimbori, Eduardo M.
; Suárez-Morales, Eduardo
; Arruda, Eliane P. de
; Chiquito, Elisandra A.
; Lima, Élison F.B.
; Castro, Elizeu B. de
; Orlandin, Elton
; Nascimento, Elynton A. do
; Razzolini, Emanuel
; Gama, Emanuel R.R.
; Araujo, Enilma M. de
; Nishiyama, Eric Y.
; Spiessberger, Erich L.
; Santos, Érika C.L. dos
; Contreras, Eugenia F.
; Galati, Eunice A.B.
; Oliveira Junior, Evaldo C. de
; Gallardo, Fabiana
; Hernandes, Fabio A.
; Lansac-Tôha, Fábio A.
; Pitombo, Fabio B.
; Dario, Fabio Di
; Santos, Fábio L. dos
; Mauro, Fabio
; Nascimento, Fabio O. do
; Olmos, Fabio
; Amaral, Fabio R.
; Schunck, Fabio
; Godoi, Fábio S. P. de
; Machado, Fabrizio M.
; Barbo, Fausto E.
; Agrain, Federico A.
; Ribeiro, Felipe B.
; Moreira, Felipe F.F.
; Barbosa, Felipe F.
; Silva, Fenanda S.
; Cavalcanti, Fernanda F.
; Straube, Fernando C.
; Carbayo, Fernando
; Carvalho Filho, Fernando
; Zanella, Fernando C.V.
; Jacinavicius, Fernando de C.
; Farache, Fernando H.A.
; Leivas, Fernando
; Dias, Fernando M.S.
; Mantellato, Fernando
; Vaz-de-Mello, Fernando Z.
; Gudin, Filipe M.
; Albuquerque, Flávio
; Molina, Flavio B.
; Passos, Flávio D.
; Shockley, Floyd W.
; Pinheiro, Francielly F.
; Mello, Francisco de A.G. de
; Nascimento, Francisco E. de L.
; Franco, Francisco L.
; Oliveira, Francisco L. de
; Melo, Francisco T. de V.
; Quijano, Freddy R.B.
; Salles, Frederico F.
; Biffi, Gabriel
; Queiroz, Gabriel C.
; Bizarro, Gabriel L.
; Hrycyna, Gabriela
; Leviski, Gabriela
; Powell, Gareth S.
; Santos, Geane B. dos
; Morse, Geoffrey E.
; Brown, George
; Mattox, George M.T.
; Zimbrão, Geraldo
; Carvalho, Gervásio S.
; Miranda, Gil F.G.
; Moraes, Gilberto J. de
; Lourido, Gilcélia M.
; Neves, Gilmar P.
; Moreira, Gilson R.P.
; Montingelli, Giovanna G.
; Maurício, Giovanni N.
; Marconato, Gláucia
; Lopez, Guilherme E.L.
; Silva, Guilherme L. da
; Muricy, Guilherme
; Brito, Guilherme R.R.
; Garbino, Guilherme S.T.
; Flores, Gustavo E.
; Graciolli, Gustavo
; Libardi, Gustavo S.
; Proctor, Heather C.
; Gil-Santana, Helcio R.
; Varella, Henrique R.
; Escalona, Hermes E.
; Schmitz, Hermes J.
; Rodrigues, Higor D.D.
; Galvão Filho, Hilton de C.
; Quintino, Hingrid Y.S.
; Pinto, Hudson A.
; Rainho, Hugo L.
; Miyahira, Igor C.
; Gonçalves, Igor de S.
; Martins, Inês X.
; Cardoso, Irene A.
; Oliveira, Ismael B. de
; Franz, Ismael
; Fernandes, Itanna O.
; Golfetti, Ivan F.
; S. Campos-Filho, Ivanklin
; Oliveira, Ivo de S.
; Delabie, Jacques H.C.
; Oliveira, Jader de
; Prando, Jadila S.
; Patton, James L.
; Bitencourt, Jamille de A.
; Silva, Janaina M.
; Santos, Jandir C.
; Arruda, Janine O.
; Valderrama, Jefferson S.
; Dalapicolla, Jeronymo
; Oliveira, Jéssica P.
; Hájek, Jiri
; Morselli, João P.
; Narita, João P.
; Martin, João P.I.
; Grazia, Jocélia
; McHugh, Joe
; Cherem, Jorge J.
; Farias Júnior, José A.S.
; Fernandes, Jose A.M.
; Pacheco, José F.
; Birindelli, José L.O.
; Rezende, José M.
; Avendaño, Jose M.
; Duarte, José M. Barbanti
; Ribeiro, José R. Inácio
; Mermudes, José R.M.
; Pujol-Luz, José R.
; Santos, Josenilson R. dos
; Câmara, Josenir T.
; Teixeira, Joyce A.
; Prado, Joyce R. do
; Botero, Juan P.
; Almeida, Julia C.
; Kohler, Julia
; Gonçalves, Julia P.
; Beneti, Julia S.
; Donahue, Julian P.
; Alvim, Juliana
; Almeida, Juliana C.
; Segadilha, Juliana L.
; Wingert, Juliana M.
; Barbosa, Julianna F.
; Ferrer, Juliano
; Santos, Juliano F. dos
; Kuabara, Kamila M.D.
; Nascimento, Karine B.
; Schoeninger, Karine
; Campião, Karla M.
; Soares, Karla
; Zilch, Kássia
; Barão, Kim R.
; Teixeira, Larissa
; Sousa, Laura D. do N.M. de
; Dumas, Leandro L.
; Vieira, Leandro M.
; Azevedo, Leonardo H.G.
; Carvalho, Leonardo S.
; Souza, Leonardo S. de
; Rocha, Leonardo S.G.
; Bernardi, Leopoldo F.O.
; Vieira, Letícia M.
; Johann, Liana
; Salvatierra, Lidianne
; Oliveira, Livia de M.
; Loureiro, Lourdes M.A. El-moor
; Barreto, Luana B.
; Barros, Luana M.
; Lecci, Lucas
; Camargos, Lucas M. de
; Lima, Lucas R.C.
; Almeida, Lucia M.
; Martins, Luciana R.
; Marinoni, Luciane
; Moura, Luciano de A.
; Lima, Luciano
; Naka, Luciano N.
; Miranda, Lucília S.
; Salik, Lucy M.
; Bezerra, Luis E.A.
; Silveira, Luis F.
; Campos, Luiz A.
; Castro, Luiz A.S. de
; Pinho, Luiz C.
; Silveira, Luiz F.L.
; Iniesta, Luiz F.M.
; Tencatt, Luiz F.C.
; Simone, Luiz R.L.
; Malabarba, Luiz R.
; Cruz, Luiza S. da
; Sekerka, Lukas
; Barros, Lurdiana D.
; Santos, Luziany Q.
; Skoracki, Maciej
; Correia, Maira A.
; Uchoa, Manoel A.
; Andrade, Manuella F.G.
; Hermes, Marcel G.
; Miranda, Marcel S.
; Araújo, Marcel S. de
; Monné, Marcela L.
; Labruna, Marcelo B.
; Santis, Marcelo D. de
; Duarte, Marcelo
; Knoff, Marcelo
; Nogueira, Marcelo
; Britto, Marcelo R. de
; Melo, Marcelo R.S. de
; Carvalho, Marcelo R. de
; Tavares, Marcelo T.
; Kitahara, Marcelo V.
; Justo, Marcia C.N.
; Botelho, Marcia J.C.
; Couri, Márcia S.
; Borges-Martins, Márcio
; Felix, Márcio
; Oliveira, Marcio L. de
; Bologna, Marco A.
; Gottschalk, Marco S.
; Tavares, Marcos D.S.
; Lhano, Marcos G.
; Bevilaqua, Marcus
; Santos, Marcus T.T.
; Domingues, Marcus V.
; Sallum, Maria A.M.
; Digiani, María C.
; Santarém, Maria C.A.
; Nascimento, Maria C. do
; Becerril, María de los A.M.
; Santos, Maria E.A. dos
; Passos, Maria I. da S. dos
; Felippe-Bauer, Maria L.
; Cherman, Mariana A.
; Terossi, Mariana
; Bartz, Marie L.C.
; Barbosa, Marina F. de C.
; Loeb, Marina V.
; Cohn-Haft, Mario
; Cupello, Mario
; Martins, Marlúcia B.
; Christofersen, Martin L.
; Bento, Matheus
; Rocha, Matheus dos S.
; Martins, Maurício L.
; Segura, Melissa O.
; Cardenas, Melissa Q.
; Duarte, Mércia E.
; Ivie, Michael A.
; Mincarone, Michael M.
; Borges, Michela
; Monné, Miguel A.
; Casagrande, Mirna M.
; Fernandez, Monica A.
; Piovesan, Mônica
; Menezes, Naércio A.
; Benaim, Natalia P.
; Reategui, Natália S.
; Pedro, Natan C.
; Pecly, Nathalia H.
; Ferreira Júnior, Nelson
; Silva Júnior, Nelson J. da
; Perioto, Nelson W.
; Hamada, Neusa
; Degallier, Nicolas
; Chao, Ning L.
; Ferla, Noeli J.
; Mielke, Olaf H.H.
; Evangelista, Olivia
; Shibatta, Oscar A.
; Oliveira, Otto M.P.
; Albornoz, Pablo C.L.
; Dellapé, Pablo M.
; Gonçalves, Pablo R.
; Shimabukuro, Paloma H.F.
; Grossi, Paschoal
; Rodrigues, Patrícia E. da S.
; Lima, Patricia O.V.
; Velazco, Paul
; Santos, Paula B. dos
; Araújo, Paula B.
; Silva, Paula K.R.
; Riccardi, Paula R.
; Garcia, Paulo C. de A.
; Passos, Paulo G.H.
; Corgosinho, Paulo H.C.
; Lucinda, Paulo
; Costa, Paulo M.S.
; Alves, Paulo P.
; Roth, Paulo R. de O.
; Coelho, Paulo R.S.
; Duarte, Paulo R.M.
; Carvalho, Pedro F. de
; Gnaspini, Pedro
; Souza-Dias, Pedro G.B.
; Linardi, Pedro M.
; Bartholomay, Pedro R.
; Demite, Peterson R.
; Bulirsch, Petr
; Boll, Piter K.
; Pereira, Rachel M.M.
; Silva, Rafael A.P.F.
; Moura, Rafael B. de
; Boldrini, Rafael
; Silva, Rafaela A. da
; Falaschi, Rafaela L.
; Cordeiro, Ralf T.S.
; Mello, Ramon J.C.L.
; Singer, Randal A.
; Querino, Ranyse B.
; Heleodoro, Raphael A.
; Castilho, Raphael de C.
; Constantino, Reginaldo
; Guedes, Reinaldo C.
; Carrenho, Renan
; Gomes, Renata S.
; Gregorin, Renato
; Machado, Renato J.P.
; Bérnils, Renato S.
; Capellari, Renato S.
; Silva, Ricardo B.
; Kawada, Ricardo
; Dias, Ricardo M.
; Siewert, Ricardo
; Brugnera, Ricaro
; Leschen, Richard A.B.
; Constantin, Robert
; Robbins, Robert
; Pinto, Roberta R.
; Reis, Roberto E. dos
; Ramos, Robson T. da C.
; Cavichioli, Rodney R.
; Barros, Rodolfo C. de
; Caires, Rodrigo A.
; Salvador, Rodrigo B.
; Marques, Rodrigo C.
; Araújo, Rodrigo C.
; Araujo, Rodrigo de O.
; Dios, Rodrigo de V.P.
; Johnsson, Rodrigo
; Feitosa, Rodrigo M.
; Hutchings, Roger W.
; Lara, Rogéria I.R.
; Rossi, Rogério V.
; Gerstmeier, Roland
; Ochoa, Ronald
; Hutchings, Rosa S.G.
; Ale-Rocha, Rosaly
; Rocha, Rosana M. da
; Tidon, Rosana
; Brito, Rosangela
; Pellens, Roseli
; Santos, Sabrina R. dos
; Santos, Sandra D. dos
; Paiva, Sandra V.
; Santos, Sandro
; Oliveira, Sarah S. de
; Costa, Sávio C.
; Gardner, Scott L.
; Leal, Sebastián A. Muñoz
; Aloquio, Sergio
; Bonecker, Sergio L.C.
; Bueno, Sergio L. de S.
; Almeida, Sérgio M. de
; Stampar, Sérgio N.
; Andena, Sérgio R.
; Posso, Sergio R.
; Lima, Sheila P.
; Gadelha, Sian de S.
; Thiengo, Silvana C.
; Cohen, Simone C.
; Brandão, Simone N.
; Rosa, Simone P.
; Ribeiro, Síria L.B.
; Letana, Sócrates D.
; Santos, Sonia B. dos
; Andrade, Sonia C.S.
; Dávila, Stephane
; Vaz, Stéphanie
; Peck, Stewart B.
; Christo, Susete W.
; Cunha, Suzan B.Z.
; Gomes, Suzete R.
; Duarte, Tácio
; Madeira-Ott, Taís
; Marques, Taísa
; Roell, Talita
; Lima, Tarcilla C. de
; Sepulveda, Tatiana A.
; Maria, Tatiana F.
; Ruschel, Tatiana P.
; Rodrigues, Thaiana
; Marinho, Thais A.
; Almeida, Thaís M. de
; Miranda, Thaís P.
; Freitas, Thales R.O.
; Pereira, Thalles P.L.
; Zacca, Thamara
; Pacheco, Thaynara L.
; Martins, Thiago F.
; Alvarenga, Thiago M.
; Carvalho, Thiago R. de
; Polizei, Thiago T.S.
; McElrath, Thomas C.
; Henry, Thomas
; Pikart, Tiago G.
; Porto, Tiago J.
; Krolow, Tiago K.
; Carvalho, Tiago P.
; Lotufo, Tito M. da C.
; Caramaschi, Ulisses
; Pinheiro, Ulisses dos S.
; Pardiñas, Ulyses F.J.
; Maia, Valéria C.
; Tavares, Valeria
; Costa, Valmir A.
; Amaral, Vanessa S. do
; Silva, Vera C.
; Wolff, Vera R. dos S.
; Slobodian, Verônica
; Silva, Vinícius B. da
; Espíndola, Vinicius C.
; Costa-Silva, Vinicius da
; Bertaco, Vinicius de A.
; Padula, Vinícius
; Ferreira, Vinicius S.
; Silva, Vitor C.P. da
; Piacentini, Vítor de Q.
; Sandoval-Gómez, Vivian E.
; Trevine, Vivian
; Sousa, Viviane R.
; Sant’Anna, Vivianne B. de
; Mathis, Wayne N.
; Souza, Wesley de O.
; Colombo, Wesley D.
; Tomaszewska, Wioletta
; Wosiacki, Wolmar B.
; Ovando, Ximena M.C.
; Leite, Yuri L.R.
.
ABSTRACT The limited temporal completeness and taxonomic accuracy of species lists, made available in a traditional manner in scientific publications, has always represented a problem. These lists are invariably limited to a few taxonomic groups and do not represent up-to-date knowledge of all species and classifications. In this context, the Brazilian megadiverse fauna is no exception, and the Catálogo Taxonômico da Fauna do Brasil (CTFB) (http://fauna.jbrj.gov.br/), made public in 2015, represents a database on biodiversity anchored on a list of valid and expertly recognized scientific names of animals in Brazil. The CTFB is updated in near real time by a team of more than 800 specialists. By January 1, 2024, the CTFB compiled 133,691 nominal species, with 125,138 that were considered valid. Most of the valid species were arthropods (82.3%, with more than 102,000 species) and chordates (7.69%, with over 11,000 species). These taxa were followed by a cluster composed of Mollusca (3,567 species), Platyhelminthes (2,292 species), Annelida (1,833 species), and Nematoda (1,447 species). All remaining groups had less than 1,000 species reported in Brazil, with Cnidaria (831 species), Porifera (628 species), Rotifera (606 species), and Bryozoa (520 species) representing those with more than 500 species. Analysis of the CTFB database can facilitate and direct efforts towards the discovery of new species in Brazil, but it is also fundamental in providing the best available list of valid nominal species to users, including those in science, health, conservation efforts, and any initiative involving animals. The importance of the CTFB is evidenced by the elevated number of citations in the scientific literature in diverse areas of biology, law, anthropology, education, forensic science, and veterinary science, among others. publications problem uptodate up date classifications context exception (CTFB http//fauna.jbrj.gov.br/, httpfaunajbrjgovbr http //fauna.jbrj.gov.br/ , jbrj gov br (http://fauna.jbrj.gov.br/) 2015 Brazil 80 specialists 1 2024 133691 133 691 133,69 125138 125 138 125,13 82.3%, 823 82 3 (82.3% 102000 102 000 102,00 7.69%, 769 7 69 (7.69% 11000 11 11,00 . 3,567 3567 567 (3,56 2,292 2292 2 292 (2,29 1,833 1833 833 (1,83 1,447 1447 447 (1,44 1000 1,00 831 (83 628 (62 606 (60 520 (52 50 users science health biology law anthropology education others http//fauna.jbrj.gov.br/ faunajbrjgovbr //fauna.jbrj.gov.br (http://fauna.jbrj.gov.br/ 201 8 202 13369 13 133,6 12513 12 125,1 82.3% (82.3 10200 10 00 102,0 7.69% 76 6 (7.69 1100 11,0 3,56 356 56 (3,5 2,29 229 29 (2,2 1,83 183 83 (1,8 1,44 144 44 (1,4 100 1,0 (8 62 (6 60 52 (5 5 http//fauna.jbrj.gov.br (http://fauna.jbrj.gov.br 20 1336 133, 1251 125, 82.3 (82. 1020 0 102, 7.69 (7.6 110 11, 3,5 35 (3, 2,2 22 (2, 1,8 18 (1, 1,4 14 4 ( 82. (82 7.6 (7. 3, (3 2, (2 (1 7. (7
7.
Development and characterization of Al2O3-based biocomposites reinforced with 3Y-TZP nanoparticles Al2O3based AlObased Al2O3 based Al O 3YTZP YTZP 3Y TZP Y AlO Al2O
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Cossu, C. M. F. A.
; Alves, M. F. R. P.
; Gomes, R. M. T.
; Strecker, K.
; Magnago, R. O.
; Santos, C.
.
Abstract Alumina ceramics were reinforced with different amounts of stabilized-tetragonal zirconia nanoparticles, 3Y-TZP, and their properties were evaluated aiming for future applications in orthopedic medicine. Different amounts of 3Y-TZP (3 to 15 wt%) were mixed with Al2O3 powder, using high-energy milling (400 rpm-24 h). Samples were uniaxially compacted and sintered at 1600 °C-2 h. The samples were characterized by their relative density, microstructure, and crystalline phases. Furthermore, Vickers hardness, fracture toughness, and bending strength were determined. After the high-energy milling process, a considerable amount of monoclinic (m) ZrO2 was detected in the powder mixtures, besides the α-Al2O3 and tetragonal (t) ZrO2 phases. After sintering the samples presented relative densities greater than 98.5%, regardless of the amount of the Y-TZP additions used. Furthermore, the monoclinic phase was reconverted into the tetragonal phase during sintering. The Vickers hardness varied between 1750 and 1690 HV, depending on the amount of Y-TZP added. Bending strength and fracture toughness were also sensitive to the addition of Y-TZP, with values increasing from 351.5 to 701.7 MPa and KIC from 3.5 to 5.6 MPa.m1/2, indicating that the t-ZrO2 grains enable the activation of the transformation toughening mechanisms such as t→m phase transformation and residual stress. The biological responses of the composites, evaluated by their cytotoxicity and chemical solubility, accredit the materials developed for future in vitro and in vivo studies aimed at application as biomaterials. stabilizedtetragonal stabilized nanoparticles 3YTZP, 3YTZP YTZP 3Y TZP, TZP Y medicine 3 ( 1 wt% wt AlO Al O Al2O highenergy high energy 400 (40 rpm24 rpm 24 rpm-2 h . h) 160 °C2 C2 C °C 2 °C- density microstructure phases Furthermore determined process m (m ZrO mixtures αAl2O3 αAlO α α-Al2O t (t 985 98 5 98.5% used 175 169 HV added YTZP, 3515 351 351. 7017 701 7 701. 35 3. 56 6 5. MPam12 MPam m1 MPa.m1/2 tZrO2 tZrO t-ZrO tm stress composites solubility biomaterials 40 (4 rpm2 rpm- 16 αAl αAl2O 9 98.5 17 70 MPam1 MPa.m1/ 4 98. MPa.m1 MPa.m
8.
Microstructure and properties of ZrO2-ZrSiO4 ceramic composites obtained by reactive sintering ZrO2ZrSiO4 ZrOZrSiO ZrO2 ZrSiO4 ZrO ZrSiO ZrO2-ZrSiO ZrO2ZrSiO
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Santanna, E. G. D.
; Gomes, P. L.
; Amarante, J. E. V.
; Alves, M. F. R. P.
; Magnago, R. O.
; Santos, C. dos
.
Abstract ZrO2-ZrSiO4 composites obtained from mixtures of 3Y-TZP and SiO2 powders were investigated. Commercial 3Y-TZP powder and mixtures containing 5 or 10 wt% of SiO2 were prepared. Specimens (n=10/group) were uniaxially compacted and sintered at 1500 °C-2 h (5 °C/min). Sintered samples were characterized by their relative density, X-ray diffraction, scanning electron microscopy, energy dispersive spectroscopy, and Vickers nanoindentation. The monolithic-ZrO2 sample presented full densification while increasing of SiO2 content progressively reduced the relative density. The crystalline phases presented in composites were tetragonal-ZrO2, cubic-ZrO2, ZrSiO4, monoclinic-ZrO2, and residual cristobalite (SiO2). Microstructural analysis indicated a distribution of zirconia grains, with heterogeneous regions rich in SiO2 surrounded by ZrSiO4 grains. Vickers hardness of 1590±19 HV for monolithic ZrO2, 1475±27 HV for ZrO2-5 wt% SiO2, and 1336±32 HV for ZrO2-10 wt% SiO2 were obtained indicating reduction in hardness with increasing SiO2 fraction. Furthermore, a reduction in fracture toughness was observed (7.2±0.8, 6.7±0.5, and 5.4±1.0 MPa.m1/2, respectively) and Young’s moduli measured were 174.1, 169.7, and 225.9 GPa, respectively. These experiments demonstrated, preliminarily, that the ZrO2-ZrSiO4 composite, based on 3Y-TZP-SiO2 powder mixtures, can achieve good levels of densification and present reasonab le mechanical properties, requiring improvements in microstructural homogenization. However, the presence of SiO2 and ZrSiO4 can improve the adhesion of zirconia to resin cement, requiring future studies focused on adhesion to confirm its viability. ZrO2ZrSiO4 ZrOZrSiO ZrO2 ZrO ZrSiO ZrO2-ZrSiO 3YTZP YTZP 3Y TZP Y SiO investigated 1 wt prepared n=10/group n10group ngroup n group (n=10/group 150 °C2 C2 C °C 2 °C- ( °C/min. Cmin °C/min . min °C/min) density Xray X ray diffraction microscopy spectroscopy nanoindentation monolithicZrO2 monolithicZrO monolithic-ZrO tetragonalZrO2, tetragonalZrO2 tetragonalZrO tetragonal tetragonal-ZrO2 cubicZrO2, cubicZrO2 cubicZrO cubic cubic-ZrO2 monoclinicZrO2, monoclinicZrO2 monoclinicZrO monoclinic monoclinic-ZrO2 SiO2. (SiO2) grains 159019 1590 19 1590±1 147527 1475 27 1475±2 ZrO25 ZrO2- 133632 1336 32 1336±3 ZrO210 ZrO2-1 fraction Furthermore 7.2±0.8, 7208 7 0 8 (7.2±0.8 6705 6 6.7±0.5 5410 4 5.4±1. MPam12 MPam MPa m1 m MPa.m1/2 respectively Youngs Young s 1741 174 174.1 1697 169 169.7 2259 225 9 225. GPa demonstrated preliminarily composite 3YTZPSiO2 YTZPSiO 3Y-TZP-SiO properties homogenization However cement viability ZrO2ZrSiO 15 tetragonal-ZrO cubic-ZrO monoclinic-ZrO (SiO2 15901 159 1590± 14752 147 1475± 13363 133 3 1336± ZrO21 7.2±0.8 720 (7.2±0. 670 6.7±0. 541 5.4±1 MPam1 MPa.m1/ 17 174. 16 169. 22 3YTZPSiO (SiO 14 13 7.2±0. 72 (7.2±0 67 6.7±0 54 5.4± MPa.m1 7.2±0 (7.2± 6.7± 5.4 MPa.m 7.2± (7.2 6.7 5. 7.2 (7. 6. 7. (7
9.
Association study between ceftriaxone and a synthetic amide against strains of Pseudomonas aeruginosa
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Rosa, L. L. S.
; Andrade-Júnior, F. P.
; Cordeiro, L. V.
; Souza, H. D. S.
; Athayde-Filho, P. F.
; Gadelha, D. D. A.
; Melo, D. M.
; Silva, D. F.
; Alves, D. N.
; Sobreira, A. L. C.
; Ferreira, S. R. D.
; Teixeira, A. P. C.
; Farias, B. K. S.
; Firmino, R. G.
; Maia, A. K. H. L.
; Lima, E. O.
.
Abstract Pseudomonas aeruginosa is a non-lactose fermenting Gram-negative bacteria responsible for causing numerous nosocomial infections. The present research aimed to analyze the anti-Pseudomonas aeruginosa potential of 2-Chloro-N-(4-fluoro-3-nitrophenyl)acetamide (A8). The antibacterial potential of A8 was evaluated from the Minimum Inhibitory Concentration (MIC), Minimum Bactericidal Concentration (MBC) and Association using the checkerboard method. MIC and MBC values were 512 µg/mL for all P. aeruginosa strains evaluated, demonstrating predominantly bactericidal activity. Furthermore, when A8 was associated with the drug ceftriaxone, pharmacological additivity and indifference were evidenced. In this sense, the synthetic amide was interesting, since it demonstrates the potential to become a possible candidate for an antimicrobial drug. nonlactose non lactose Gramnegative Gram negative infections antiPseudomonas anti 2ChloroN4fluoro3nitrophenylacetamide ChloroNfluoronitrophenylacetamide 2 Chloro N 4 fluoro 3 nitrophenyl acetamide A8. A . (A8) MIC, , (MIC) (MBC method 51 µgmL µg mL P activity Furthermore ceftriaxone evidenced sense interesting ChloroN nitrophenylacetamide (A8 (MIC 5 (A
Resumo Pseudomonas aeruginosa é uma bactéria Gram-negativa não fermentadora de lactose, responsável por causar inúmeras infecções nosocomiais. A presente pesquisa teve como objetivo analisar o potencial anti-Pseudomonas aeruginosa da molécula 2-Cloro-N-(4-fluoro-3-nitrofenil)acetamida (A8). O potencial antibacteriano do A8 foi avaliado a partir da Concentração Inibitória Mínima (CIM), Concentração Bactericida Mínima (CBM) e Associação pelo método de checkboard. Os valores de CIM e CBM foram de 512 µg/mL para todas as cepas de P. aeruginosa avaliadas, demonstrando atividade predominantemente bactericida. Além disso, quando o A8 foi associado ao fármaco ceftriaxona, evidenciou-se aditividade e indiferença farmacológica. Nesse sentido, a amida sintética se mostrou interessante, pois demonstra potencial para se tornar um possível candidato a fármaco antimicrobiano. Gramnegativa Gram negativa lactose nosocomiais antiPseudomonas anti 2CloroN4fluoro3nitrofenilacetamida CloroNfluoronitrofenilacetamida 2 Cloro N 4 fluoro 3 nitrofenil acetamida A8. . (A8) CIM, , (CIM) (CBM checkboard 51 µgmL µg mL P avaliadas bactericida disso ceftriaxona evidenciouse evidenciou farmacológica sentido interessante antimicrobiano CloroN nitrofenilacetamida (A8 (CIM 5 (A
10.
Racial and economic segregation in Brazil: a nationwide analysis of socioeconomic and socio-spatial inequalities Brazil sociospatial socio spatial
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Sousa Filho, José Firmino de
; Pedeira, Sara Costa
; Santos, Gervásio F. dos
; Guimarães, Joanna M. N.
; Ferreira, Andrêa J. F.
; Alves, Flávia Jôse O.
; Nascimento, Gabrielle R.
; Paiva, Aureliano S. S.
; Andrade, Roberto F. S.
; Góes, Emanuelle F.
; Barreto, Maurício L.
; Aquino, Estela M. L.
.
Resumen Este artículo tiene como objetivo analizar la segregación residencial por raza (segregación racial) y renta (segregación económica) en Brasil y explorar su relación con factores socioeconómicos y socioespaciales. La segregación residencial se evaluó utilizando el índice de disimilitud con base en el censo demográfico de 2010 y considerando las secciones censales urbanas ya que la segregación es considerada sociológicamente como un problema urbano. Los resultados para la segregación racial mostraron que esta es más evidente en ciudades del sur y del sudeste de Brasil y que afecta principalmente a la población autodeclarada negra. El enfoque usado para calcular la segregación económica implicó examinar el nivel de ingresos de diferentes grupos de bajos ingresos. Por lo tanto, consideramos que las familias que ganaban entre cero y un salario mínimo son el grupo con mayor vulnerabilidad social. No encontramos correlaciones significativas entre los índices de segregación racial y los de ingresos con factores como la urbanización (tamaño de la población urbana). Finalmente, presentamos los índices de segregación racial estratificando a las familias por umbrales de renta para las 27 capitales brasileñas y concluimos que la renta per cápita de los hogares es un factor preponderante para la segregación de los más pobres, en especial en las familias cuyos habitantes se autodeclaran negros. socioespaciales 201 urbano negra tanto social tamaño urbana. urbana . urbana) Finalmente 2 pobres negros 20
Abstract This article aims to analyze residential segregation by race (racial segregation) and income (economic segregation) in Brazil and explore its relationship with socioeconomic and socio-spatial factors. Residential segregation was assessed using the dissimilarity index based on the 2010 demographic census and considering urban census tracts since segregation is sociologically considered an urban problem. The results for racial segregation showed that it is more evident in cities in the South and Southeast of Brazil and mainly affects the self-declared black population. The approach used to calculate economic segregation involved examining the income level of different low-income groups. Therefore, we consider families that earned between 0 and 1 minimum wage as the group with the greatest social vulnerability. We did not find significant correlations between racial and income segregation indices with aspects such as urbanization (urban population size). Finally, we present the racial segregation indices stratifying families by income thresholds for the 27 Brazilian capitals and conclude that per capita household income is a preponderant factor for the segregation of the poorest, especially in families whose residents self-identify as black. sociospatial socio spatial factors 201 problem selfdeclared self declared lowincome low groups Therefore vulnerability size. size . size) Finally 2 poorest selfidentify identify 20
Resumo Este artigo tem como objetivo analisar a segregação residencial por raça (segregação racial) e renda (segregação econômica) no Brasil e explorar sua relação com fatores socioeconômicos e socioespaciais. A segregação residencial foi avaliada pelo índice de dissimilaridade baseado no Censo Demográfico de 2010 e considerando setores censitários urbanos, uma vez que a segregação é entendida sociologicamente como um problema urbano. Os resultados mostram que a segregação racial é mais evidente nas cidades do Sul e Sudeste do Brasil, atingindo principalmente a população autodeclarada preta. A abordagem utilizada para calcular a segregação econômica envolveu examinar o nível de renda de diferentes grupos de baixa renda. Portanto, consideramos as famílias que ganham entre 0 e 1 salário mínimo - o grupo de maior vulnerabilidade social. Não encontramos correlações significativas entre os índices de segregação racial e de renda com fatores como a urbanização (tamanho da população urbana). Por fim, apresentamos os índices de segregação racial estratificando as famílias por faixas de renda para as 27 capitais brasileiras e concluímos que a renda domiciliar per capita é fator preponderante para a segregação dos mais pobres, principalmente nas famílias cujos moradores se autodeclaram pretos. socioespaciais 201 urbanos urbano preta Portanto social tamanho urbana. urbana . urbana) fim 2 pobres pretos 20
11.
In vitro Antioxidant and Anticholinesterase Activities of Ouratea fieldingiana (Gardner) Eng. Leaf Extract and Correlation with Its Phenolics Profile with an in silico Study in Relation to Alzheimer’s Disease
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Frota, Lucas S.
; Alves, Daniela R.
; Freitas, Leonardo S.
; Lopes, Francisco F. S.
; Marinho, Marcia M.
; Marinho, Emmanuel S.
; Morais, Selene M. de
.
Journal of the Brazilian Chemical Society
- Métricas do periódico
Ouratea fieldingiana is a native medicinal plant from Northeastern Brazil and many biological properties are due to the phenolic constituents. The objective of this work was performing the characterization of O. fieldingiana leaf constituents to correlate with antioxidant and anticholinesterase activities by in vitro and in silico studies and thus contribute to find new agents against Alzheimer’s disease. The high-performance liquid chromatography revealed the presence of the flavonoids rutin, isoquercitrin, kaempferol-3-O-rutinoside, quercetin, apigenin and amentoflavone. The antioxidant activities by the (2,2-diphenyl-1-picrylhydrazyl) (DPPH) and 2,2’-azino-bis(3-ethylbenzothiazoline-6-sulfonic acid) (ABTS) methodologies, showed good results with half maximal inhibitory concentration (IC50) values ranging from 5.63 to 11.47 µg mL-1 and 2.72 to 23.71 µg mL-1, respectively. Acetylcholinesterase inhibition assay pointed out the flavone apigenin with best activity. Computational studies evaluated the interaction of flavonoids with the enzyme acetylcholinesterase co-crystallized with the galantamine, used as standard. All flavonoids exhibited binding energy greater than that of galantamine, but only apigenin showed strong interaction with the active site of the enzyme and other bind probably to different allosteric centers. Then, O. fieldingiana extract and flavonoids with good anti-radical activity and presenting a broad-spectrum action against acetylcholinesterase (AChE) enzyme ought to be tested in clinical studies to discover new neuro-therapeutic candidates.
12.
Protein-coding gene interaction network prediction of bioactive plant compound action against SARS-CoV-2: a novel hypothesis using bioinformatics analysis
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SANTOS SOBRINHO, ELIANE M.
; SANTOS, HÉRCULES O.
; MARTINS, ERNANE R.
; FONSECA, FRANCINE SOUZA ALVES DA
; FARIAS, LUCYANA C.
; AGUILAR, CHARLES M.
; PEREIRA, ULISSES A.
; NICOLAU JUNIOR, NILSON
; GOMES, MATHEUS S.
; SOUZA, CINTYA N. DE
; RAVNJAK, JOÃO MATHEUS A.
; PORTO, RAPHAEL R.
; ALMEIDA, ANNA CHRISTINA DE
.
Abstract This study aimed to verify the action of bioactive compounds from Brazilian plants on the leader genes involved in the SARS-CoV-2 pathway. The main human genes involved were identified in GeneCards and UNIPROT platforms, and an interaction network between leader genes was established in the STRING database. To design chemo-biology interactome networks and elucidate the interplay between genes related to the disease and bioactive plant compounds, the metasearch engine STITCH 3.1 was used. The analysis revealed that SMAD3 and CASP3 genes are leader genes, suggesting that the mechanism of action of the virus on host cells is associated with the molecular effects of these genes. Furthermore, the bioactive plant compounds, such as ascorbate, benzoquinone, ellagic acid, and resveratrol was identified as a promising adjuvant for the treatment inhibiting CASP3-mediated apoptosis. Bioactive plant compounds were verified as the main pathways enriched with KEGG and related to viral infection, assessments/immune/infections, and cell proliferation, which are potentially used for respiratory viral infections. The best-ranked molecule docked in the CASP3 binding site was rutin, while the SMAD3 binding site was resveratrol. In conclusion, this work identified several bioactive compounds from Brazilian plants showing potential antiviral functions that can directly or indirectly inhibit the new coronavirus.
13.
A first approximation for the Herpetofauna species composition of the Taiamã Ecological Station, Pantanal of Mato Grosso, Brazil
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Silva-Alves, V. D.
; Mudrek, J. R.
; Silva-Diogo, O.
; Canale, G. R.
; Santos-Filho, M.
; Muniz, C. C.
; Silva, D. J.
.
14.
Shelf Life of Bioactive Compounds from Acerola Pulp (Malpighia spp.) through Freeze-Drying and Microencapsulation
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Saqueti, Bruno H. F.
; Alves, Eloize S.
; Castro, Matheus C.
; Santos, Patrícia D. S. dos
; Sinosaki, Nayane B. M.
; Senes, Carlos E. R.
; Visentainer, Jesuí V.
; Santos, Oscar O.
.
Journal of the Brazilian Chemical Society
- Métricas do periódico
Acerola is a tropical fruit with a large industrial and commercial appeal due to its organoleptic qualities and bioactive compound-rich nature. Thus, as bioactive compounds (BC) stability is of great interest in the food industry, assessment of preserving techniques to prolong shelf life has become imperative. Hence, the purpose of this study was to evaluate how storage affects BC conservation in microencapsulated and lyophilized acerola pulps over 180 days. For this matter, antioxidant tests, physical-chemical analyzes, and vitamin C analysis by mass spectrometry were performed. Results indicated that microencapsulation better preserved the antioxidants in acerola pulp compared to the other preservation technologies employed. This is due to the greater BC concentration in the microencapsulated, as well as the pH reduction. Furthermore, over 180 days, microencapsulation better preserved the target compounds in acerola pulp compared to lyophilization, as evidenced by the superior content of BC in the former treatment, making it an appealing option for the food sector.
https://doi.org/10.21577/0103-5053.20210096
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15.
A Systematic Pipeline to Enhance the Fecal Metabolome Coverage by LC-HRMS
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Alves, Marina A.
; Silva, Ana Carolina R. da
; Torres, Clarisse L.
; Almeida, Lana R. de
; Mastella, Ana Maria O.
; Borges, Ricardo M.
; Garrett, Rafael
.
Journal of the Brazilian Chemical Society
- Métricas do periódico
The comprehended knowledge of the metabolic profile of the fecal matter has been recognized as an important point for understanding metabolic changes in the human systemic metabolism and it can provide precious information about host-gut microbiota interactions. However, few analytical strategies have been addressed for a broad analysis of metabolites with different chemical properties to better understand the chemical space of fecal samples. Here we report a systematic pipeline to achieve comprehensive coverage of the fecal metabolome, from high polar to nonpolar metabolites, using dog fecal samples as a proof-of-concept. This pipeline comprises a monophasic (ACN/H2O) and a biphasic extraction (methyl tert-butyl ether (MTBE)/MeOH/H2O) of the sample, followed by three liquid chromatography-high resolution tandem mass spectrometry (LC-HRMS/MS) methods using HILIC-amide, RP-C18 and CSH-C18 columns, and a switch polarity acquisition mode in the electrospray ion source. This approach allowed the annotation of 376 metabolites from 70 different chemical classes. The chemical space analysis by molecular networking and the pathway analysis revealed the complexity of the fecal sample and the importance of combined methods to better understand biochemical pathways. This pipeline can be used as a valuable tool to comprehend the relationship between host-gut microbiota metabolites and the influence of diet, medication, or environmental changes.
https://doi.org/10.21577/0103-5053.20210042
108 downloads
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